Benzenesulfonamide

Benzenesulfonamide

SCHEMBL3603399

NS(=O)(=O)c1ccccc1.c1ccc(N2CO2)cc1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 17/20 0.59
CA2 P00918 17/20 0.59
CA12 O43570 14/20 0.59
CA9 Q16790 14/20 0.59
CA7 P43166 4/20 0.59
CA14 Q9ULX7 3/20 0.59
CA4 P22748 2/20 0.59
CA3 P07451 1/20 0.59
CA6 P23280 1/20 0.59
CA5A P35218 1/20 0.59
PLA2G7 Q13093 1/20 0.59
CA13 Q8N1Q1 1/20 0.59
CA5B Q9Y2D0 1/20 0.59
PTGS1 P23219 2/20 0.44
PTGS2 P35354 2/20 0.44
SOS1 Q07889 1/20 0.43
SCN2A Q99250 1/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1406399 0.79
Benzenesulfonamide SCHEMBL729 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
SCHEMBL19479299 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL6868390 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL1332409 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL28257999 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL29825137 0.77 CA2 (1.00) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL1009443 0.75 CA2 (0.94) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL3056735 0.75 CA2 (0.94) CA1CA2CA12CA9CA7
Benzenesulfonamide SCHEMBL3100364 0.75 CA2 (0.94) CA1CA2CA12CA9CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8541475-B2 MAO-B inhibitors useful for treating obesity JENRIN DISCOVERY, INC. (US) 2013-09-24 US disclosed
CN-101300006-B MAO-B inhibitors useful for treating obesity DISCOVERY JENRIN 2012-07-25 CN disclosed
US-20100168068-A1 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2010-07-01 US disclosed
US-7649115-B2 MAO-B inhibitors useful for treating obesity JENRIN DISCOVERY, INC. (US) 2010-01-19 US disclosed
CN-101300006-A MAO-B inhibitors useful for treating abesity DISCOVERY JENRIN (US) 2008-11-05 CN disclosed
EP-1890690-A2 MAO-B INHIBITORS USEFUL FOR TREATING ABESITY Jenrin Discovery (US) 2008-02-27 EP disclosed
US-20070088004-A1 Monoamine oxidase-B inhibitors; , and/or cardiometabolic disorders ( hypertension, dyslipidemias, high blood pressure, and insulin resistance); JENRIN DISCOVERY, INC. 2007-04-19 US disclosed
WO-2006130707-A2 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2006-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070088004-A1 Monoamine oxidase-B inhibitors; , and/or cardiometabolic disorders ( hypertension, dyslipidemias, high blood pressure, and insulin resistance); MAOB, MAOA, APOB CA1 4838/4885CA2 3532/4885CA12 4764/4885
US-20100168068-A1 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY MAOB, MAOA, GPR119 CA1 4802/4885CA2 3637/4885CA12 4773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.