SCHEMBL360405

SCHEMBL360405

COc1ccc(-n2ncc(C(=O)NC3CCN(C)C3)c2C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
PKM P14618 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 2/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
CHRNB2 P17787 2/20 0.47
CHRNA4 P43681 2/20 0.47
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD11B1 P28845 1/20 0.47
CTSL P07711 1/20 0.47
CTSS P25774 1/20 0.47
CTSK P43235 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL360081 1.00 NPC1 (0.53) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL3395172 0.79 NPC1 (0.56) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL3392885 0.79 NPC1 (0.56) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL2927664 0.76 CTSL (0.58) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL12931786 0.74 MAPT (0.55) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL3395175 0.73 SPR (0.62) NPC1RAB9APKMKMT2AMEN1
SCHEMBL3392887 0.73 SPR (0.62) NPC1RAB9APKMKMT2AMEN1
SCHEMBL10364511 0.73 HSD11B1 (0.53) NPC1RAB9ASMN1; SMN2MAPTKMT2A
SCHEMBL2855932 0.73 NPC1 (0.69) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL2857152 0.72 NPC1 (0.91) NPC1RAB9APKMSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed