SCHEMBL3607622

SCHEMBL3607622

N#Cc1cc(C(N)=O)sc1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
ALDH1A1 P00352 3/20 0.39
SLC9A1 P19634 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CDK8 P49336 2/20 0.35
ICAM1 P05362 2/20 0.35
SELE P16581 2/20 0.35
VCAM1 P19320 2/20 0.35
F2 P00734 1/20 0.35
CCNC P24863 1/20 0.35
KDR P35968 2/20 0.34
DAPK3 O43293 2/20 0.34
CSNK1A1 P48729 2/20 0.34
LIMK1 P53667 2/20 0.34
ROCK1 Q13464 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
DYRK1B Q9Y463 2/20 0.34
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3609749 0.90 GAA (0.36) GAAALDH1A1SLC9A1NPSR1L3MBTL1
SCHEMBL3605972 0.74 NOTUM (0.43) ALDH1A1KDM4EMAPTNOTUM
SCHEMBL4211782 0.69 KDR (0.43) GAAALDH1A1CDK8ICAM1SELE
SCHEMBL31117978 0.69 SLC9A1 (0.72) SLC9A1CDK8ICAM1SELEVCAM1
SCHEMBL12272939 0.69 ALDH1A1 (0.46) GAAALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL29684344 0.67 SIRT2 (0.39) GAAALDH1A1SLC9A1CDK8ICAM1
SCHEMBL3610681 0.65 KDM4E (0.42) GAAALDH1A1L3MBTL1KDRCSNK2A2
SCHEMBL21788571 0.65 LIMK1 (0.47) GAAALDH1A1SLC9A1NPSR1LIMK1
SCHEMBL29684490 0.64 F2 (0.34) CDK8ICAM1SELEVCAM1F2
SCHEMBL29684364 0.64 NOTUM (0.39) CDK8ICAM1SELEVCAM1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835476-B2 Synthesis of novel antimicrobials WU FAN (CA) 2014-09-16 US disclosed
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials WU FAN 2010-03-25 US disclosed
WO-2006092059-A1 DESIGN AND SYNTHESIS OF NOVEL ANTIMICROBIALS WU FAN (CA) 2006-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials MLX, LPXN, TPX2 GAA 1273/4885ALDH1A1 4295/4885SLC9A1 2480/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.