SCHEMBL3615591

SCHEMBL3615591

CC(C)N(C(=O)N1CCN(c2nc(N)nc3sc(-c4ccc(F)cc4)cc23)CC1)C(C)C.Nc1nc(N2CCC(C(=O)c3ccccc3)CC2)c2cc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.46
GPR55 Q9Y2T6 1/20 0.42
P2RY12 Q9H244 5/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CNR1 P21554 2/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD11B1 P28845 3/20 0.39
STAT3 P40763 3/20 0.39
HRH4 Q9H3N8 2/20 0.39
CYP2D6 P10635 1/20 0.38
NR2F2 P24468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653372 0.91 CNR2 (0.48) CNR2GPR55P2RY12KDM4EALDH1A1
SCHEMBL655170 0.90 CNR2 (0.48) CNR2GPR55KDM4EALDH1A1CNR1
SCHEMBL653833 0.77 ALDH1A1 (0.52) CNR2GPR55KDM4EALDH1A1CNR1
SCHEMBL656257 0.75 GFER (0.53) CNR2GPR55P2RY12KDM4EALDH1A1
SCHEMBL655251 0.75 L3MBTL1 (0.46) CNR2GPR55P2RY12KDM4EALDH1A1
SCHEMBL654795 0.74 ENPP2 (0.52) CNR2GPR55P2RY12KDM4EALDH1A1
SCHEMBL3621794 0.74 TP53 (0.46) CNR2GPR55KDM4EALDH1A1CNR1
SCHEMBL653429 0.72 PI4KB (0.62) CNR2GPR55P2RY12ALDH1A1
SCHEMBL794422 0.72 HRH4 (0.46) CNR2KDM4EALDH1A1CNR1HPGD
SCHEMBL653760 0.71 KDM4E (0.50) CNR2GPR55KDM4EALDH1A1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010103130-A2 NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-09-16 WO disclosed