SCHEMBL361734

SCHEMBL361734

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
KIF11 P52732 1/20 0.33
BRD4 O60885 2/20 0.33
LMNA P02545 3/20 0.32
KDM4E B2RXH2 2/20 0.32
IDH1 O75874 2/20 0.32
GPR27 Q9NS67 1/20 0.32
CNR2 P34972 1/20 0.31
ADRB2 P07550 2/20 0.31
ADRB1 P08588 2/20 0.31
ADRB3 P13945 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
EP300 Q09472 1/20 0.31
GLA P06280 1/20 0.30
BLM P54132 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362297 0.88 MGAM (0.38) SLC6A2SLC6A4SLC6A3KCNH2KIF11
SCHEMBL365294 0.86 GPBAR1 (0.35) GPBAR1BRD4KDM4EMEN1KMT2A
SCHEMBL365274 0.85 GPBAR1 (0.46) GPBAR1SLC6A3BRD4MEN1KMT2A
SCHEMBL363288 0.83 GPBAR1 (0.39) GPBAR1KDM4EMEN1KMT2AEP300
SCHEMBL12505651 0.83 GPBAR1 (0.35) GPBAR1BRD4
SCHEMBL363112 0.83 GPBAR1 (0.36) GPBAR1BRD4
SCHEMBL363178 0.83 GPBAR1 (0.51) GPBAR1BRD4ADRB1ADRB3MEN1
SCHEMBL1389707 0.82 GPBAR1 (0.37) GPBAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL369952 0.82 GPBAR1 (0.37) GPBAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL362795 0.81 GPBAR1 (0.36) GPBAR1SLC6A3BRD4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed