SCHEMBL362081

SCHEMBL362081

CC(=O)[C@](c1ccc(O)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.33
HSD17B2 P37059 1/20 0.33
NR3C2 P08235 1/20 0.32
SORT1 Q99523 1/20 0.31
ESR1 P03372 2/20 0.30
ESR2 Q92731 2/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363061 0.91 KCNN4 (0.34) NR3C2SORT1
SCHEMBL364193 0.89 NPC1 (0.34) NR3C2SORT1ALDH1A1CYP3A4
SCHEMBL363549 0.89 NPC1 (0.34) NR3C2SORT1ALDH1A1CYP3A4
SCHEMBL363211 0.89 NPC1 (0.34) NR3C2SORT1ALDH1A1CYP3A4
SCHEMBL365152 0.87 PTPN1 (0.33) NR3C2
SCHEMBL363769 0.87 PTPN1 (0.33) NR3C2
SCHEMBL363020 0.86 ATR (0.35) ALDH1A1
SCHEMBL363805 0.85 GPBAR1 (0.31)
SCHEMBL364263 0.85 GPBAR1 (0.31)
SCHEMBL363702 0.85 NPC1 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed