SCHEMBL363211

SCHEMBL363211

CC(=O)C(c1ccc(Br)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SORT1 Q99523 3/20 0.34
TRPV1 Q8NER1 1/20 0.33
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
NR3C2 P08235 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MAPT P10636 3/20 0.31
KDM4E B2RXH2 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
CASP3 P42574 1/20 0.30
SENP8 Q96LD8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363549 1.00 NPC1 (0.34) NPC1RAB9ASORT1TRPV1TP53
SCHEMBL364193 1.00 NPC1 (0.34) NPC1RAB9ASORT1TRPV1TP53
SCHEMBL363061 0.90 KCNN4 (0.34) SORT1MAPK1NR3C2NPSR1KDM4E
SCHEMBL362720 0.89 SORT1 (0.33) NPC1RAB9ASORT1NR3C2ALDH1A1
SCHEMBL362081 0.89 HSD17B1 (0.33) SORT1NR3C2ALDH1A1CYP3A4
SCHEMBL364536 0.88 SORT1 (0.35) SORT1TRPV1ALDH1A1CYP1A2CYP3A4
SCHEMBL364659 0.86 KCNK3 (0.33) NPC1RAB9ASORT1TRPV1ALDH1A1
SCHEMBL363769 0.86 PTPN1 (0.33) NR3C2
SCHEMBL364539 0.86 POLB (0.32)
SCHEMBL365152 0.86 PTPN1 (0.33) NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed