SCHEMBL363020

SCHEMBL363020

CC(=O)[C@](c1ccc(S(C)(=O)=O)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.35
MAPK14 Q16539 1/20 0.34
PTGS2 P35354 5/20 0.33
PTGS1 P23219 1/20 0.33
GRM5 P41594 1/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
MAP4K4 O95819 1/20 0.32
TGFBR1 P36897 1/20 0.32
ALDH1A1 P00352 2/20 0.32
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364667 0.90 NR1H2 (0.42) ATRMAPK14PTGS2NR1H2NR1H3
SCHEMBL363246 0.88 NR1H2 (0.33) ATRMAPK14PTGS2PTGS1GRM5
SCHEMBL363061 0.87 KCNN4 (0.34) KDM5AKDM4CKDM5B
SCHEMBL362081 0.86 HSD17B1 (0.33) ALDH1A1
SCHEMBL363457 0.86 CCR9 (0.38) ATRMAPK14PTGS2PTGS1
SCHEMBL363211 0.85 NPC1 (0.34) ALDH1A1
SCHEMBL363549 0.85 NPC1 (0.34) ALDH1A1
SCHEMBL364193 0.85 NPC1 (0.34) ALDH1A1
SCHEMBL363769 0.83 PTPN1 (0.33)
SCHEMBL365152 0.83 PTPN1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed