SCHEMBL363702

SCHEMBL363702

CCOc1ccc([C@@](C(C)=O)(c2ccnc(C)c2)c2ccccc2C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.39
RAB9A P51151 5/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
PKM P14618 3/20 0.39
TP53 P04637 3/20 0.37
LMNA P02545 3/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 3/20 0.36
MITF O75030 1/20 0.36
KMT2A Q03164 4/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
BCL2 P10415 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362932 0.87 RAB9A (0.33) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL364004 0.86 MAPT (0.41) NPC1RAB9ASMN1; SMN2PKMTP53
SCHEMBL363061 0.86 KCNN4 (0.34) KDM4EEDNRBEDNRANPSR1
SCHEMBL362081 0.85 HSD17B1 (0.33) ALDH1A1
SCHEMBL363769 0.84 PTPN1 (0.33)
SCHEMBL365152 0.84 PTPN1 (0.33)
SCHEMBL363549 0.84 NPC1 (0.34) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL364193 0.84 NPC1 (0.34) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL363211 0.84 NPC1 (0.34) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL364143 0.82 FFAR1 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed