SCHEMBL3624947

SCHEMBL3624947

N#Cc1cc(F)c(NC2CCC(NC(=O)O)CC2)nc1Cl

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.46
KHK P50053 1/20 0.42
PDE4B Q07343 7/20 0.38
PDE4D Q08499 6/20 0.38
PDE4A P27815 5/20 0.38
PDE4C Q08493 5/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
IRAK4 Q9NWZ3 2/20 0.37
HPGD P15428 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3624945 1.00 ACHE (0.46) ACHEKHKPDE4BPDE4DPDE4A
SCHEMBL17498356 0.89 KHK (0.51) ACHEKHKROCK2ROCK1IRAK4
SCHEMBL3630702 0.88 ACHE (0.47) ACHEIRAK4KMT2A
SCHEMBL3630704 0.88 ACHE (0.47) ACHEIRAK4KMT2A
SCHEMBL3630458 0.85 KDM4E (0.41) ACHEPDE4BPDE4DPDE4APDE4C
SCHEMBL3630454 0.85 KDM4E (0.41) ACHEPDE4BPDE4DPDE4APDE4C
SCHEMBL9107040 0.85 KHK (0.41) ACHEKHK
SCHEMBL14911459 0.85 KHK (0.41) ACHEKHK
SCHEMBL2713345 0.85 KHK (0.41) ACHEKHK
SCHEMBL3628370 0.83 ROCK2 (0.53) PDE4BPDE4DPDE4APDE4CROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010032875-A2 HETEROCYCLIC CARBOXAMIDE COMPOUNDS ASTELLAS PHARMA INC. (JP) 2010-03-25 WO disclosed