SCHEMBL3628240

SCHEMBL3628240

Cc1nccc2nc(C(N)CCN3CCN(C)CC3)ccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
SLC2A1 P11166 1/20 0.33
HRH3 Q9Y5N1 2/20 0.32
HRH4 Q9H3N8 1/20 0.32
OGA O60502 1/20 0.32
CYP3A4 P08684 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD3 P35462 1/20 0.32
OPRK1 P41145 1/20 0.32
PDE4D Q08499 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDE3A Q14432 1/20 0.32
HTR3A P46098 1/20 0.32
USP2 O75604 2/20 0.31
ACHE P22303 1/20 0.31
SRC P12931 1/20 0.31
CYP2D6 P10635 1/20 0.31
CCR5 P51681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3630469 0.79 HRH3 (0.38) KDM4ESLC2A1HRH3KCNH2
SCHEMBL3633564 0.79 CYP2C9 (0.45) ACHENOS3NOS1
SCHEMBL3320336 0.74 MEN1 (0.52) DRD3KCNH2NOS3NOS1NOS2
SCHEMBL3321404 0.73 MEN1 (0.45) ALDH1A1KDM4EHRH3DRD3
SCHEMBL3631614 0.72 LMNA (0.37) HRH3KCNH2
SCHEMBL3322526 0.71 NMT1 (0.48) SLC2A1HRH3HRH4ACHESRC
SCHEMBL3633491 0.71 LPAR2 (0.43) ALDH1A1KDM4E
SCHEMBL3663850 0.68 SIGMAR1 (0.45)
SCHEMBL3317233 0.65 MEN1 (0.50) HRH3
SCHEMBL3321913 0.64 MEN1 (0.49) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP disclosed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO disclosed