SCHEMBL362932

SCHEMBL362932

CCOc1ccc([C@@](C(C)=NO)(c2ccnc(C)c2)c2ccccc2C)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.33
NPC1 O15118 4/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
PKM P14618 2/20 0.33
GPBAR1 Q8TDU6 2/20 0.33
TP53 P04637 3/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
ADORA2A P29274 1/20 0.32
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 2/20 0.31
KIF11 P52732 1/20 0.31
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
ESR1 P03372 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CHRNB2 P17787 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363702 0.87 NPC1 (0.39) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL364569 0.87 MAPT (0.36) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL364180 0.86 GPBAR1 (0.35) GPBAR1
SCHEMBL364263 0.85 GPBAR1 (0.31) GPBAR1
SCHEMBL363805 0.85 GPBAR1 (0.31) GPBAR1
SCHEMBL364217 0.85 GPBAR1 (0.30) GPBAR1
SCHEMBL364539 0.84 POLB (0.32) GPBAR1
SCHEMBL364836 0.84 POLB (0.32) GPBAR1
SCHEMBL362228 0.82 ALDH1A1 (0.31)
SCHEMBL363246 0.81 NR1H2 (0.33) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed