SCHEMBL363246

SCHEMBL363246

CC(=NO)[C@](c1ccc(S(C)(=O)=O)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.33
MAP4K4 O95819 1/20 0.32
TGFBR1 P36897 1/20 0.32
MAPK14 Q16539 1/20 0.32
GRM5 P41594 1/20 0.32
ATR Q13535 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.31
NR1H3 Q13133 2/20 0.31
PTGS2 P35354 5/20 0.31
ALOX5 P09917 1/20 0.30
SYK P43405 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365085 0.91 NR1H2 (0.41) NR1H2MAP4K4TGFBR1MAPK14ATR
SCHEMBL364292 0.91 NR1H2 (0.34) NR1H2GRM5GPBAR1NR1H3
SCHEMBL363020 0.88 ATR (0.35) NR1H2MAP4K4TGFBR1MAPK14GRM5
SCHEMBL363922 0.88 NR1H2 (0.41) NR1H2MAP4K4NR1H3PTGS2SYK
SCHEMBL363868 0.87 CCR9 (0.34) MAPK14GRM5ATRPTGS2PTGS1
SCHEMBL365288 0.87 CCR9 (0.34) MAPK14GRM5ATRPTGS2PTGS1
SCHEMBL364180 0.86 GPBAR1 (0.35) GPBAR1
SCHEMBL364263 0.85 GPBAR1 (0.31) GPBAR1
SCHEMBL363805 0.85 GPBAR1 (0.31) GPBAR1
SCHEMBL364539 0.84 POLB (0.32) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed