SCHEMBL3630587

SCHEMBL3630587

CC(C)(O)CNS(=O)(=O)c1ccccc1C=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.44
ALOX5AP P20292 2/20 0.42
FEN1 P39748 2/20 0.42
ELANE P08246 1/20 0.38
PRTN3 P24158 1/20 0.38
CA12 O43570 6/20 0.37
CA9 Q16790 6/20 0.37
CYP2C9 P11712 1/20 0.37
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
THRB P10828 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NEK1 Q96PY6 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993438 0.80 CA12 (0.44) CYP2C19ALOX5APFEN1CA12CA9
SCHEMBL15915560 0.78 RECQL (0.55) CYP2C19ALOX5APFEN1CA12CA9
SCHEMBL20267870 0.78 GBA1 (0.54) CYP2C19ALOX5APFEN1MEN1KMT2A
SCHEMBL2801003 0.76 ALDH1A1 (0.44) CYP2C19ALOX5APFEN1CYP2C9MEN1
SCHEMBL2801005 0.75 NSD2 (0.47) CYP2C19ALOX5APFEN1ELANEPRTN3
SCHEMBL11890046 0.75 CYP2C19 (0.73) CYP2C19CA12CA9LMNAALDH1A1
SCHEMBL2798389 0.74 LMNA (0.46) CYP2C19ELANEPRTN3CYP2C9MEN1
SCHEMBL7184559 0.74 CA1 (0.52) CYP2C19ELANEPRTN3CYP2C9MEN1
SCHEMBL2799637 0.74 CA12 (0.58) CA12CA9LMNAKMT2AALDH1A1
SCHEMBL14398993 0.74 PKLR (0.49) CA12CA9LMNATHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148862-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. Hoffmann-Roche AG (CH) 2010-02-03 EP disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed