SCHEMBL363066

SCHEMBL363066

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NC[C@@H](O)CO)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.35
BRD4 O60885 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HRH1 P35367 4/20 0.33
CCR3 P51677 4/20 0.33
MAPK14 Q16539 2/20 0.32
GCGR P47871 2/20 0.32
KCNH2 Q12809 1/20 0.32
KDR P35968 4/20 0.32
TP53 P04637 1/20 0.32
EPHX2 P34913 1/20 0.32
PYGL P06737 1/20 0.31
GCG P01275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363811 0.93 S1PR1 (0.36) GPBAR1BRD4KDM4EALDH1A1HPGD
SCHEMBL362795 0.89 GPBAR1 (0.36) GPBAR1BRD4ALDH1A1HPGDGCGR
SCHEMBL362902 0.89 GPBAR1 (0.45) GPBAR1BRD4KDM4EALDH1A1HPGD
SCHEMBL363289 0.86 GPBAR1 (0.41) GPBAR1BRD4KDM4EALDH1A1HPGD
SCHEMBL365274 0.85 GPBAR1 (0.46) GPBAR1BRD4
SCHEMBL363112 0.85 GPBAR1 (0.36) GPBAR1BRD4ALDH1A1GCGRTP53
SCHEMBL362887 0.84 GPBAR1 (0.39) GPBAR1BRD4ALDH1A1HPGDTP53
SCHEMBL369578 0.84 GPBAR1 (0.35) GPBAR1BRD4KDM4EALDH1A1HPGD
SCHEMBL369576 0.84 GPBAR1 (0.35) GPBAR1BRD4KDM4EALDH1A1HPGD
SCHEMBL369579 0.84 GPBAR1 (0.35) GPBAR1BRD4KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed