SCHEMBL3632208

SCHEMBL3632208

O=C(O)c1c2cc(=O)cc(F)c-2cn(-c2ccccc2)c1CBr

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 3/20 0.33
LMNA P02545 1/20 0.32
COMT P21964 1/20 0.32
RORC P51449 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632440 0.85 MAPK1 (0.40) MAPK1KDM4ELMNACOMTRORC
SCHEMBL4316385 0.81 MEN1 (0.43) MAPK1KDM4ELMNACOMTALDH1A1
SCHEMBL3625416 0.80 KDM4E (0.34) MAPK1KDM4ECOMTALDH1A1
SCHEMBL3632144 0.75 ABCB1 (0.37) KDM4ELMNA
SCHEMBL3634031 0.73 PLA2G4A (0.35) MAPK1
SCHEMBL3632665 0.72 ABCB1 (0.50) KDM4ELMNAALDH1A1HPGD
SCHEMBL3633358 0.72 NOTUM (0.44) KDM4ELMNAALDH1A1
SCHEMBL3634622 0.72 NOTUM (0.45) KDM4ELMNA
SCHEMBL3631523 0.71 MAPK1 (0.38) MAPK1KDM4ELMNARORC
SCHEMBL3635017 0.71 GABRA2 (0.36) MAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed