SCHEMBL3632144

SCHEMBL3632144

O=C(O)c1c2cc(=O)ccc-2cn(-c2ccc(F)cc2)c1CBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.37
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
METTL3 Q86U44 2/20 0.33
METTL14 Q9HCE5 2/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
CHRNA7 P36544 2/20 0.33
BCL2L1 Q07817 1/20 0.32
BAD Q92934 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
TP53 P04637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ATM Q13315 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3625416 0.89 KDM4E (0.34) KDM4EGABRA2GABRB2NOTUMMAPT
SCHEMBL3633608 0.81 ABCB1 (0.53) ABCB1LMNAKDM4EGABRA2GABRB2
SCHEMBL3635017 0.81 GABRA2 (0.36) KDM4EGABRA2GABRB2KMT2AMEN1
SCHEMBL3628060 0.81 ALKBH5 (0.37) LMNAKDM4EKMT2AMEN1TP53
SCHEMBL3631576 0.77 ALDH1A1 (0.35) LMNAKDM4EKMT2AMEN1ATM
SCHEMBL3634602 0.77 NR4A3 (0.37) KDM4EGABRA2GABRB2
SCHEMBL3632208 0.75 MAPK1 (0.35) LMNAKDM4E
SCHEMBL3627357 0.74 ALDH1A1 (0.35) LMNAKDM4EATMMAPT
SCHEMBL3627548 0.74 COMT (0.33) LMNAKDM4EGABRA2GABRB2KMT2A
SCHEMBL3634680 0.74 GRIA1 (0.35) LMNAKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed