SCHEMBL365085

SCHEMBL365085

CC(=NO)C(c1cccc(-c2ccc(S(C)(=O)=O)cc2)c1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.41
MAPK14 Q16539 1/20 0.38
SYK P43405 1/20 0.37
NR1H3 Q13133 4/20 0.37
CYP2C9 P11712 1/20 0.36
MAP4K4 O95819 3/20 0.35
TGFBR1 P36897 3/20 0.35
PTGS2 P35354 3/20 0.34
LRRK2 Q5S007 2/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
RXRA P19793 1/20 0.34
PTGS1 P23219 1/20 0.33
ATR Q13535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363246 0.91 NR1H2 (0.33) NR1H2MAPK14SYKNR1H3MAP4K4
SCHEMBL364667 0.90 NR1H2 (0.42) NR1H2MAPK14SYKNR1H3CYP2C9
SCHEMBL364292 0.90 NR1H2 (0.34) NR1H2NR1H3LRRK2RXRA
SCHEMBL363922 0.83 NR1H2 (0.41) NR1H2SYKNR1H3MAP4K4PTGS2
SCHEMBL364180 0.82 GPBAR1 (0.35)
SCHEMBL363020 0.79 ATR (0.35) NR1H2MAPK14NR1H3MAP4K4TGFBR1
SCHEMBL364971 0.79 GPBAR1 (0.31)
SCHEMBL365288 0.78 CCR9 (0.34) MAPK14PTGS2PTGS1ATR
SCHEMBL363868 0.78 CCR9 (0.34) MAPK14PTGS2PTGS1ATR
SCHEMBL364263 0.77 GPBAR1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed