SCHEMBL363922

SCHEMBL363922

C/C(=N/O)C(c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1)(c1ccnc(C)c1)c1ccccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.41
KIF11 P52732 1/20 0.40
PTGS2 P35354 5/20 0.38
PTGS1 P23219 2/20 0.38
SYK P43405 1/20 0.38
NR1H3 Q13133 4/20 0.37
CYP2D6 P10635 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
MAP4K4 O95819 1/20 0.37
PIK3CA P42336 1/20 0.37
KCNH2 Q12809 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
RORC P51449 1/20 0.37
FLT3 P36888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363246 0.88 NR1H2 (0.33) NR1H2PTGS2PTGS1SYKNR1H3
SCHEMBL365085 0.83 NR1H2 (0.41) NR1H2PTGS2PTGS1SYKNR1H3
SCHEMBL364311 0.83 POLB (0.31) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL362574 0.81 SYK (0.40) SYKRORC
SCHEMBL365421 0.79 NR1H2 (0.39) NR1H2KIF11PTGS2PTGS1SYK
SCHEMBL363868 0.79 CCR9 (0.34) PTGS2PTGS1CYP2D6PSEN1PSEN2
SCHEMBL365288 0.79 CCR9 (0.34) PTGS2PTGS1CYP2D6PSEN1PSEN2
SCHEMBL364292 0.79 NR1H2 (0.34) NR1H2KIF11NR1H3CYP2D6PSEN1
SCHEMBL364334 0.77 NR1H2 (0.41) NR1H2KIF11PTGS2PTGS1SYK
SCHEMBL363020 0.76 ATR (0.35) NR1H2PTGS2PTGS1NR1H3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed