SCHEMBL3633378

SCHEMBL3633378

CCC(Nc1ccc2c(C)nccc2n1)C1CCCN1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
BACE1 P56817 1/20 0.33
SLC6A2 P23975 6/20 0.32
SLC6A3 Q01959 6/20 0.32
SLC6A4 P31645 5/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835204 0.72 NR4A2 (0.55) BACE1PDE3AMEN1KMT2A
SCHEMBL19477394 0.68 SLC6A2 (0.37) SLC6A2SLC6A3SLC6A4
SCHEMBL3225927 0.67 MEN1 (0.41) BACE1SLC6A2SLC6A3SLC6A4MEN1
SCHEMBL3971157 0.66 PDE5A (0.35)
SCHEMBL7441662 0.64 HTR3A (0.33) SLC6A2SLC6A3SLC6A4
SCHEMBL3327779 0.63 PRKCD (0.48)
SCHEMBL3321416 0.63 ACHE (0.54) KMT2A
SCHEMBL3320135 0.62 NMT1 (0.48)
SCHEMBL3321755 0.62 HRH3 (0.47)
SCHEMBL3322501 0.61 ALDH1A1 (0.55) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP disclosed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO disclosed