SCHEMBL363349

SCHEMBL363349

Cc1ccccc1[C@@H](C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.66
BRD4 O60885 1/20 0.39
MGAM O43451 2/20 0.34
GAA P10253 2/20 0.34
SI P14410 2/20 0.34
MGAM2 Q2M2H8 2/20 0.34
CTSA P10619 2/20 0.34
CHEK2 O96017 1/20 0.34
RXRA P19793 4/20 0.33
RXRB P28702 4/20 0.33
RXRG P48443 1/20 0.33
MLKL Q8NB16 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
GRIK1 P39086 1/20 0.32
GRIK2 Q13002 1/20 0.32
GRIK3 Q13003 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362545 1.00 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL364601 1.00 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL363678 0.97 GPBAR1 (0.61) GPBAR1BRD4MGAMGAASI
SCHEMBL363650 0.93 GPBAR1 (0.58) GPBAR1BRD4MGAMGAASI
SCHEMBL362527 0.92 GPBAR1 (0.55) GPBAR1BRD4MGAMGAASI
SCHEMBL363444 0.92 GPBAR1 (0.55) GPBAR1BRD4MGAMGAASI
SCHEMBL362317 0.88 GPBAR1 (0.52) GPBAR1BRD4CTSA
SCHEMBL361842 0.88 GPBAR1 (0.51) GPBAR1BRD4CTSARXRARXRB
SCHEMBL361676 0.88 GPBAR1 (0.51) GPBAR1BRD4CTSARXRARXRB
SCHEMBL371037 0.88 GPBAR1 (0.49) GPBAR1BRD4MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed