SCHEMBL361676

SCHEMBL361676

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(CCC(=O)O)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.51
FFAR1 O14842 10/20 0.39
BRD4 O60885 1/20 0.36
FFAR4 Q5NUL3 4/20 0.34
CHRM2 P08172 1/20 0.34
S1PR1 P21453 1/20 0.34
FPR1 P21462 1/20 0.34
FPR3 P25089 1/20 0.34
GPR183 P32249 1/20 0.34
APLNR P35414 1/20 0.34
GPR65 Q8IYL9 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
CTSA P10619 1/20 0.33
LMNA P02545 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
MMEL1 Q495T6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362545 0.88 GPBAR1 (0.66) GPBAR1BRD4RXRARXRBRXRG
SCHEMBL364092 0.88 GPBAR1 (0.48) GPBAR1FFAR1BRD4CTSALMNA
SCHEMBL363349 0.88 GPBAR1 (0.66) GPBAR1BRD4RXRARXRBRXRG
SCHEMBL364601 0.88 GPBAR1 (0.66) GPBAR1BRD4RXRARXRBRXRG
SCHEMBL363650 0.85 GPBAR1 (0.58) GPBAR1BRD4RXRARXRBRXRG
SCHEMBL363678 0.85 GPBAR1 (0.61) GPBAR1BRD4CTSA
SCHEMBL362317 0.84 GPBAR1 (0.52) GPBAR1FFAR1BRD4S1PR1CTSA
SCHEMBL364071 0.83 GPBAR1 (0.47) GPBAR1BRD4
SCHEMBL363585 0.82 GPBAR1 (0.45) GPBAR1BRD4
SCHEMBL362350 0.81 GPBAR1 (0.48) GPBAR1BRD4CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed