SCHEMBL363444

SCHEMBL363444

Cc1cc(/C(CC(c2ccc(-c3ccc(C(=O)O)cc3)cc2)c2ccccc2F)=N/O)c[nH]c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.55
BRD4 O60885 1/20 0.37
TTR P02766 1/20 0.34
RXRA P19793 3/20 0.34
HNF4A P41235 1/20 0.34
MGAM O43451 2/20 0.33
GAA P10253 2/20 0.33
SI P14410 2/20 0.33
MGAM2 Q2M2H8 2/20 0.33
HDAC4 P56524 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
RXRB P28702 2/20 0.32
RXRG P48443 1/20 0.32
CTSA P10619 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362545 0.92 GPBAR1 (0.66) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL364601 0.92 GPBAR1 (0.66) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL363349 0.92 GPBAR1 (0.66) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL362457 0.90 GPBAR1 (0.48) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL362281 0.90 GPBAR1 (0.48) GPBAR1BRD4RXRAHNF4ARXRB
SCHEMBL362527 0.89 GPBAR1 (0.55) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL363678 0.88 GPBAR1 (0.61) GPBAR1BRD4TTRMGAMGAA
SCHEMBL361680 0.88 GPBAR1 (0.47) GPBAR1BRD4RXRAMGAMGAA
SCHEMBL361842 0.87 GPBAR1 (0.51) GPBAR1BRD4TTRRXRARXRB
SCHEMBL363235 0.87 GPBAR1 (0.51) GPBAR1BRD4RXRAHNF4ARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed