SCHEMBL363650

SCHEMBL363650

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2cccc(C(=O)O)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.58
KMO O15229 1/20 0.38
BRD4 O60885 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
GAA P10253 2/20 0.35
LMNA P02545 1/20 0.35
CTSA P10619 2/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
MGAM O43451 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
TDP2 O95551 1/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364601 0.93 GPBAR1 (0.66) GPBAR1BRD4GAACTSAMGAM
SCHEMBL363349 0.93 GPBAR1 (0.66) GPBAR1BRD4GAACTSAMGAM
SCHEMBL362545 0.93 GPBAR1 (0.66) GPBAR1BRD4GAACTSAMGAM
SCHEMBL363678 0.90 GPBAR1 (0.61) GPBAR1BRD4GAACTSAMGAM
SCHEMBL362317 0.88 GPBAR1 (0.52) GPBAR1BRD4CTSA
SCHEMBL361676 0.85 GPBAR1 (0.51) GPBAR1BRD4LMNACTSARXRA
SCHEMBL363444 0.85 GPBAR1 (0.55) GPBAR1BRD4GAACTSAMGAM
SCHEMBL362527 0.85 GPBAR1 (0.55) GPBAR1BRD4GAACTSAMGAM
SCHEMBL364092 0.84 GPBAR1 (0.48) GPBAR1BRD4GAALMNACTSA
SCHEMBL361842 0.84 GPBAR1 (0.51) GPBAR1BRD4LMNACTSARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed