SCHEMBL3634102

SCHEMBL3634102

Cc1c[nH]c(-c2ccc(N)cc2OC(C)C)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK9 P50750 1/20 0.36
CCNA1 P78396 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
TLR8 Q9NR97 1/20 0.35
PDE7A Q13946 3/20 0.33
PDE7B Q9NP56 2/20 0.33
PDE4D Q08499 1/20 0.33
MCHR1 Q99705 1/20 0.33
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
PDE5A O76074 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
CASP6 P55212 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1967098 0.84 IMPDH2 (0.44) PDE7APDE7BPDE4DALDH1A1GAA
SCHEMBL3663746 0.77 ALDH1A1 (0.41) ALDH1A1GAAKDM4ELMNAPOLB
SCHEMBL3733422 0.75 PDE5A (0.31) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL3660492 0.75 CYP3A4 (0.43) ALDH1A1GAAKDM4ELMNAPOLB
SCHEMBL3411515 0.75 KIT (0.37) PDE7AALDH1A1GAAKDM4ELMNA
SCHEMBL3633331 0.71 KDM4E (0.41) ALDH1A1KDM4ELMNAMCL1MDM4
SCHEMBL3637473 0.69 IMPDH2 (0.43) PDE7APDE7BPDE4DALDH1A1GAA
SCHEMBL1226779 0.69 PDE7A (0.44) PDE7APDE7BPDE4DALDH1A1GAA
SCHEMBL6747997 0.68 IMPDH2 (0.42) TLR8MCHR1ALDH1A1GAAIMPDH2
SCHEMBL8145073 0.68 ALDH1A1 (0.48) TLR8MCHR1ALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed