SCHEMBL3663746

SCHEMBL3663746

Cc1c[nH]c(-c2ccc(N)cc2C)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
PDE10A Q9Y233 1/20 0.37
KDM4E B2RXH2 5/20 0.37
MAPT P10636 5/20 0.37
GAA P10253 4/20 0.37
HPGD P15428 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
RECQL P46063 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 3/20 0.37
LMNA P02545 2/20 0.37
CASP6 P55212 1/20 0.37
CASP1 P29466 2/20 0.35
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
THRB P10828 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660492 0.83 CYP3A4 (0.43) ALDH1A1KDM4EMAPTGAAHPGD
SCHEMBL3411515 0.83 KIT (0.37) ALDH1A1KDM4EMAPTGAAHPGD
SCHEMBL1967098 0.81 IMPDH2 (0.44) ALDH1A1KDM4EMAPTGAALMNA
SCHEMBL3633331 0.80 KDM4E (0.41) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL3634102 0.77 CCNT1 (0.36) ALDH1A1KDM4EGAAPOLBLMNA
SCHEMBL24360032 0.74 DCUN1D1 (0.50) ALDH1A1KDM4EGAAHPGDNPC1
SCHEMBL3635215 0.74 NPC1 (0.44) ALDH1A1KDM4EMAPTGAAHPGD
SCHEMBL15651168 0.74 NISCH (0.46) ALDH1A1PDE10AKDM4EMAPTGAA
SCHEMBL6802067 0.72 HPGD (0.50) ALDH1A1KDM4EMAPTGAAHPGD
SCHEMBL16280579 0.72 ALDH1A1 (0.65) ALDH1A1PDE10AKDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed
WO-2008137102-A2 METHODS OF MODULATING AMYLOID BETA AND COMPOUNDS USEFUL THEREFOR TORREYPINES THERAPEUTICS, INC. (US) 2008-11-13 WO disclosed