SCHEMBL3634836

SCHEMBL3634836

CC1CN(C[CH]c2ccc3cnccc3n2)CCN1CCCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.45
OPRM1 P35372 1/20 0.37
HTR1A P08908 2/20 0.36
SLC6A4 P31645 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3320692 0.81 SIGMAR1 (0.44) SIGMAR1OPRM1HTR1A
SCHEMBL3663846 0.71 SIGMAR1 (0.47) SIGMAR1
SCHEMBL14645859 0.71 SIGMAR1 (0.68) SIGMAR1
SCHEMBL10998697 0.59 LMNA (0.49) SIGMAR1OPRM1HTR1ASLC6A4
SCHEMBL4169559 0.59 SIGMAR1 (0.67) SIGMAR1
SCHEMBL11789571 0.58 SIGMAR1 (0.62) SIGMAR1
SCHEMBL1309373 0.58 HRH2 (0.52) SIGMAR1
Bromide SCHEMBL4174825 0.58 SIGMAR1 (0.65) SIGMAR1
SCHEMBL29748826 0.58 SIGMAR1 (0.52) SIGMAR1
SCHEMBL28283654 0.58 CHRNB2 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP disclosed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO disclosed