SCHEMBL3663846

SCHEMBL3663846

Cc1nccc2nc([CH]CN3CCN(CCCc4ccccc4)CC3)ccc12

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.47
POLB P06746 1/20 0.45
LTA4H P09960 1/20 0.41
GRIN2B Q13224 1/20 0.41
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632725 0.87 ACHE (0.44) SIGMAR1GRIN2B
SCHEMBL3633456 0.79 HRH3 (0.38)
SCHEMBL3320690 0.79 SIGMAR1 (0.47) SIGMAR1POLBGRIN2B
SCHEMBL3663850 0.77 SIGMAR1 (0.45) SIGMAR1POLBGRIN2BCYP2C9
SCHEMBL3322228 0.72 ACHE (0.47) SIGMAR1CYP2C9
SCHEMBL3627515 0.71 KDM4E (0.37)
SCHEMBL3632511 0.71 KDM2B (0.42)
SCHEMBL3633564 0.70 CYP2C9 (0.45) CYP2C9
SCHEMBL3320215 0.69 CARM1 (0.48) SIGMAR1GRIN2B
SCHEMBL6550825 0.68 SIGMAR1 (1.00) SIGMAR1POLBLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP disclosed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO disclosed