SCHEMBL363623

SCHEMBL363623

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(Oc2cccc(C(=O)O)c2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.39
AKR1C3 P42330 1/20 0.37
PPARG P37231 7/20 0.37
KDR P35968 2/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
CYP2C9 P11712 1/20 0.35
RAB9A P51151 1/20 0.35
KMO O15229 1/20 0.34
FLT1 P17948 1/20 0.33
FABP1 P07148 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363688 0.91 GPBAR1 (0.38) GPBAR1MRGPRX4POLB
SCHEMBL369888 0.89 KDR (0.38) GPBAR1AKR1C3PPARGKDRMRGPRX4
SCHEMBL362892 0.86 GPBAR1 (0.39) GPBAR1
SCHEMBL361842 0.84 GPBAR1 (0.51) GPBAR1
SCHEMBL1390092 0.83 GPBAR1 (0.40) GPBAR1AKR1C3PPARGMRGPRX4
SCHEMBL1390090 0.83 GPBAR1 (0.40) GPBAR1AKR1C3PPARGMRGPRX4
SCHEMBL363245 0.81 GPBAR1 (0.43) GPBAR1
SCHEMBL365756 0.81 ADRB3 (0.38) GPBAR1AKR1C3PPARGMRGPRX4NPC1
SCHEMBL363831 0.80 GPBAR1 (0.42) GPBAR1PPARGCYP2C9
SCHEMBL363394 0.79 MRGPRX4 (0.40) GPBAR1PPARGKDRMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed