SCHEMBL363394

SCHEMBL363394

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(Oc2cccc(C(=O)O)c2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.40
PTGER4 P35408 2/20 0.37
PTGER2 P43116 1/20 0.37
PPARG P37231 4/20 0.34
KDR P35968 2/20 0.34
GPBAR1 Q8TDU6 2/20 0.34
P2RX3 P56373 2/20 0.33
IDO1 P14902 1/20 0.33
NR4A2 P43354 1/20 0.33
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365756 0.89 ADRB3 (0.38) MRGPRX4PPARGGPBAR1P2RX3NR4A2
SCHEMBL363129 0.89 FFAR1 (0.34) MRGPRX4PTGER4PTGER2KDRGPBAR1
SCHEMBL362921 0.85 MRGPRX4 (0.40) MRGPRX4PTGER4PTGER2PPARGGPBAR1
SCHEMBL362920 0.85 MRGPRX4 (0.40) MRGPRX4PTGER4PTGER2PPARGGPBAR1
SCHEMBL362499 0.83 PPARG (0.32) PPARGGPBAR1
SCHEMBL364251 0.83 MEN1 (0.35) GPBAR1
SCHEMBL363628 0.82 ADRB1 (0.35) PTGER4PTGER2KDRGPBAR1P2RX3
SCHEMBL369888 0.82 KDR (0.38) MRGPRX4PPARGKDRGPBAR1P2RX3
SCHEMBL365274 0.81 GPBAR1 (0.46) MRGPRX4GPBAR1
SCHEMBL363178 0.79 GPBAR1 (0.51) PPARGGPBAR1ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed