SCHEMBL365756

SCHEMBL365756

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(Oc2cccc(C(=O)O)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 4/20 0.38
GPBAR1 Q8TDU6 2/20 0.38
MRGPRX4 Q96LA9 2/20 0.38
KMO O15229 1/20 0.37
AKR1C3 P42330 1/20 0.36
ADRB1 P08588 2/20 0.36
POLB P06746 2/20 0.36
PPARG P37231 1/20 0.36
NPC1 O15118 1/20 0.36
CYP2C9 P11712 1/20 0.36
RAB9A P51151 1/20 0.36
P2RX3 P56373 5/20 0.36
NR4A2 P43354 1/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
SNCA P37840 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363394 0.89 MRGPRX4 (0.40) ADRB3GPBAR1MRGPRX4ADRB1PPARG
SCHEMBL370059 0.89 GPBAR1 (0.35) ADRB3GPBAR1ADRB1P2RX3
SCHEMBL363628 0.88 ADRB1 (0.35) ADRB3GPBAR1ADRB1POLBP2RX3
SCHEMBL365274 0.87 GPBAR1 (0.46) GPBAR1MRGPRX4POLBMEN1KMT2A
SCHEMBL369888 0.85 KDR (0.38) GPBAR1MRGPRX4AKR1C3POLBPPARG
SCHEMBL363178 0.85 GPBAR1 (0.51) ADRB3GPBAR1ADRB1POLBPPARG
SCHEMBL364384 0.83 P2RX3 (0.41) ADRB3GPBAR1MRGPRX4KMOPOLB
SCHEMBL364385 0.83 P2RX3 (0.41) ADRB3GPBAR1MRGPRX4KMOPOLB
SCHEMBL362064 0.82 CNR1 (0.37) GPBAR1POLBPPARG
SCHEMBL363623 0.81 GPBAR1 (0.39) GPBAR1MRGPRX4KMOAKR1C3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed