SCHEMBL3636451

SCHEMBL3636451

O=c1[nH]c2ccccc2n1C1CCN(C[C@@H]2CCCN2Cc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 11/20 0.72
OPRK1 P41145 2/20 0.72
OPRL1 P41146 2/20 0.72
DRD4 P21917 1/20 0.56
AKT1 P31749 1/20 0.56
AKT2 P31751 1/20 0.56
AKT3 Q9Y243 1/20 0.56
PLD1 Q13393 1/20 0.55
ALDH1A1 P00352 2/20 0.55
KDM4E B2RXH2 1/20 0.55
PMP22 Q01453 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
TSHR P16473 1/20 0.55
MAPK1 P28482 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637576 0.97 OPRM1 (0.71) OPRM1OPRK1OPRL1DRD4AKT1
SCHEMBL3665096 0.84 OPRM1 (1.00) OPRM1OPRK1OPRL1DRD4AKT1
SCHEMBL3758854 0.83 OPRM1 (0.52) OPRM1OPRK1OPRL1ALDH1A1KDM4E
Oxalic Acid SCHEMBL5778025 0.82 OPRM1 (0.91) OPRM1OPRK1OPRL1DRD4AKT1
SCHEMBL3751742 0.82 CHRM2 (0.60) OPRM1OPRK1OPRL1ALDH1A1KDM4E
SCHEMBL3751747 0.82 CHRM2 (0.60) OPRM1OPRK1OPRL1ALDH1A1KDM4E
SCHEMBL8863557 0.80 OPRM1 (0.91) OPRM1OPRK1OPRL1DRD4AKT1
SCHEMBL11223608 0.80 OPRM1 (0.86) OPRM1OPRK1OPRL1DRD4AKT1
SCHEMBL4679567 0.80 OPRM1 (0.55) OPRM1OPRK1OPRL1ALDH1A1KDM4E
SCHEMBL4679560 0.80 OPRM1 (0.55) OPRM1OPRK1OPRL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP disclosed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO disclosed