SCHEMBL3636604

SCHEMBL3636604

O=C(O)c1cccc(F)c1Nc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.54
MEN1 O00255 4/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
CXCR2 P25025 2/20 0.53
ALB P02768 1/20 0.52
FABP4 P15090 1/20 0.51
MAPT P10636 2/20 0.49
DHODH Q02127 1/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 2/20 0.46
CDC7 O00311 1/20 0.46
AURKA O14965 1/20 0.46
MAPK8 P45983 1/20 0.46
ALK Q9UM73 1/20 0.46
ALOX15 P16050 1/20 0.45
GFER P55789 1/20 0.45
NGLY1 Q96IV0 1/20 0.45
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8285642 0.87 CXCR2 (0.60) KMT2AMEN1CXCR2FABP4MAPT
SCHEMBL28289321 0.84 KDM4E (0.64) KMT2AMEN1NPC1RAB9ACXCR2
SCHEMBL3364068 0.82 POLB (0.60) KMT2AMEN1CXCR2FABP4MAPT
SCHEMBL15698772 0.81 MAP2K1 (0.56) KMT2AMEN1NPC1RAB9ACXCR2
SCHEMBL2406195 0.81 MAPT (0.62) KMT2AMEN1CXCR2FABP4MAPT
SCHEMBL21312751 0.80 KMT2A (0.53) KMT2AMEN1NPC1RAB9AMAPT
SCHEMBL29220911 0.80 FABP4 (0.68) KMT2AMEN1CXCR2FABP4MAPT
SCHEMBL7573159 0.79 CXCR2 (0.47) KMT2AMEN1CXCR2ALBALDH1A1
SCHEMBL24021598 0.79 CLCN2 (0.61) KMT2AMEN1ALBFABP4MAPT
SCHEMBL11542345 0.79 CXCR2 (0.53) KMT2AMEN1CXCR2FABP4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9946847-B2 Libraries of compounds having desired properties and methods for making and using them BIOBLOCKS INC. (US) 2018-04-17 US disclosed
US-20150269356-A1 LIBRARIES OF COMPOUNDS HAVING DESIRED PROPERTIES AND METHODS FOR MAKING AND USING THEM BIOBLOCKS INC (US) 2015-09-24 US disclosed
US-20150269356-A1 LIBRARIES OF COMPOUNDS HAVING DESIRED PROPERTIES AND METHODS FOR MAKING AND USING THEM BIOBLOCKS INC (US) 2015-09-24 US disclosed
WO-2014047463-A2 LIBRARIES OF COMPOUNDS HAVING DESIRED PROPERTIES AND METHODS FOR MAKING AND USING THEM BIOBLOCKS, INC. (US) 2014-03-27 WO disclosed
EP-2148862-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. Hoffmann-Roche AG (CH) 2010-02-03 EP disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed
US-4168312-A Quinolone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-09-18 US disclosed