SCHEMBL3636997

SCHEMBL3636997

COC(=O)c1[nH]c2cc(C)ccc2c(=O)c1Cc1ccc2c(c1)OCO2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.51
KDM4E B2RXH2 8/20 0.51
HSD17B10 Q99714 6/20 0.51
POLB P06746 3/20 0.51
USP2 O75604 3/20 0.51
LMNA P02545 1/20 0.51
MEN1 O00255 6/20 0.49
KMT2A Q03164 6/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MAPT P10636 5/20 0.48
HTT P42858 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 3/20 0.45
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3938675 0.87 HSD17B10 (0.47) ALDH1A1KDM4EHSD17B10POLBUSP2
SCHEMBL3635425 0.77 HPGD (0.42) ALDH1A1KDM4EHSD17B10USP2MEN1
SCHEMBL9281684 0.75 HTT (0.59) ALDH1A1KDM4EHSD17B10USP2MEN1
SCHEMBL3630797 0.75 EDNRB (0.41) ALDH1A1KDM4EHSD17B10POLBUSP2
SCHEMBL3634856 0.70 PTGS1 (0.46) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL847034 0.69 SMN1; SMN2 (0.52) ALDH1A1KDM4EHSD17B10USP2LMNA
SCHEMBL13856579 0.68 ALDH1A1 (1.00) ALDH1A1KDM4EHSD17B10POLBUSP2
SCHEMBL848642 0.67 MAPK8 (0.59) KDM4EMEN1KMT2ATSHR
SCHEMBL3634795 0.67 MAPK8 (0.42) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL20272215 0.66 RGS12 (0.58) ALDH1A1KDM4EHSD17B10POLBUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148862-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. Hoffmann-Roche AG (CH) 2010-02-03 EP disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed