SCHEMBL3637649

SCHEMBL3637649

CC(=O)Nc1ccc2c(c1)nc(C(=O)O)n2C(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.53
KDM4E B2RXH2 8/20 0.50
MAPT P10636 6/20 0.50
RAB9A P51151 6/20 0.50
ALDH1A1 P00352 4/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
GLA P06280 1/20 0.50
TNNI3 P19429 1/20 0.50
TNNT2 P45379 1/20 0.50
TNNC1 P63316 1/20 0.50
RUNX1 Q01196 1/20 0.50
CBFB Q13951 1/20 0.50
PABPC1 P11940 1/20 0.48
POLB P06746 1/20 0.47
GFER P55789 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.44
ACSS2 Q9NR19 1/20 0.44
LDHA P00338 1/20 0.44
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637823 0.79 ALOX5AP (0.43) KDM4EALDH1A1TDP1
SCHEMBL4072935 0.70 NPC1 (0.44) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL617991 0.69 NPC1 (1.00) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL18075701 0.68 KDM4E (1.00) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL6965384 0.68 RAB9A (0.46) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL22930416 0.67 MAPT (1.00) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL26802185 0.67 RAB9A (0.68) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL11055398 0.67 MAPT (0.56) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL10347621 0.66 MAPT (0.55) NPC1KDM4EMAPTRAB9AALDH1A1
SCHEMBL3731059 0.66 NPC1 (0.55) NPC1KDM4EMAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed