SCHEMBL3637823

SCHEMBL3637823

CC(C)(C)n1c(C(=O)O)nc2cc(N)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 9/20 0.43
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 3/20 0.39
CHEK1 O14757 2/20 0.39
AURKA O14965 2/20 0.39
CSNK1A1 P48729 2/20 0.39
LIMK1 P53667 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
DAPK3 O43293 1/20 0.39
GSK3A P49840 1/20 0.39
IKBKE Q14164 1/20 0.39
MAPK14 Q16539 1/20 0.39
TAOK1 Q7L7X3 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
RAD52 P43351 1/20 0.39
HTT P42858 1/20 0.39
HCAR3 P49019 1/20 0.38
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637649 0.79 NPC1 (0.53) ALDH1A1KDM4ETDP1
SCHEMBL28693493 0.77 NR1H2 (0.41) ALDH1A1KDM4ECHEK1AURKACSNK1A1
SCHEMBL8045718 0.73 CCR2 (0.47) ALOX5APALDH1A1KDM4ECHEK1AURKA
SCHEMBL15544534 0.71 KDM4E (0.46) ALDH1A1KDM4ECHEK1AURKACSNK1A1
SCHEMBL482647 0.71 ALDH1A1 (0.41) ALOX5APALDH1A1KDM4ECHEK1AURKA
SCHEMBL6420483 0.70 KDM4E (0.45) KDM4ECHEK1AURKACSNK1A1LIMK1
SCHEMBL28681187 0.69 GABRG2 (0.41) ALDH1A1KDM4ECHEK1AURKACSNK1A1
SCHEMBL335868 0.67 NPC1 (0.47) ALDH1A1KDM4ECHEK1AURKACSNK1A1
SCHEMBL14000394 0.65 ALDH1A1 (0.70) ALDH1A1KDM4EHTT
SCHEMBL2364886 0.65 PKM (0.44) KDM4EDYRK1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed