SCHEMBL3640646

SCHEMBL3640646

O=C(NCC[C]1CC1)c1cccc2occc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MAOB P27338 1/20 0.40
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
THRB P10828 1/20 0.40
MRGPRX1 Q96LB2 1/20 0.40
HCRTR1 O43613 5/20 0.39
HCRTR2 O43614 4/20 0.39
HPGD P15428 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3647326 0.82 HPGD (0.44) MTNR1AMTNR1BMAOBALDH1A1SMN1; SMN2
SCHEMBL3647331 0.82 MAOB (0.59) MTNR1AMTNR1BMAOBALDH1A1NPC1
SCHEMBL3645922 0.81 MAOB (0.45) MTNR1AMTNR1BMAOBALDH1A1NPC1
SCHEMBL3640648 0.80 MAOB (0.48) MAOBNPC1RAB9AMRGPRX1HCRTR1
SCHEMBL3647212 0.80 MTNR1A (0.47) MTNR1AMTNR1BMAOBALDH1A1NPC1
SCHEMBL3646928 0.80 MTNR1A (0.50) MTNR1AMTNR1BMAOBNPC1RAB9A
SCHEMBL3645919 0.80 MAOB (0.41) MTNR1AMTNR1BMAOBMRGPRX1HCRTR1
SCHEMBL3645101 0.80 LMNA (0.48) MAOBNPC1RAB9ASMN1; SMN2MRGPRX1
SCHEMBL3641406 0.79 MRGPRX1 (0.46) MTNR1AMTNR1BMAOBMRGPRX1HCRTR1
SCHEMBL3641411 0.79 MRGPRX1 (0.46) ALDH1A1SMN1; SMN2MRGPRX1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188282-A2 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2010-05-26 EP disclosed
WO-2009022311-A2 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2009-02-19 WO disclosed