SCHEMBL3645989

SCHEMBL3645989

CC(C)(C)C(Cc1cc(S(=O)(=O)c2cccnc2)c(-c2cccnc2Cl)s1)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
KCNJ8 Q15842 1/20 0.35
MCL1 Q07820 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
NAMPT P43490 5/20 0.33
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ADAM17 P78536 1/20 0.31
MAPT P10636 1/20 0.31
TBXAS1 P24557 1/20 0.31
DHODH Q02127 1/20 0.31
CYP2C9 P11712 1/20 0.31
PIK3CD O00329 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653192 0.90 ABCC9 (0.36) ABCC9ABCC8KCNJ11KCNJ8GPBAR1
SCHEMBL3648437 0.88 GPBAR1 (0.36) ABCC9ABCC8KCNJ11KCNJ8MCL1
SCHEMBL3654495 0.87 ABCC9 (0.37) ABCC9ABCC8KCNJ11KCNJ8GPBAR1
SCHEMBL3649651 0.82 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8NAMPT
SCHEMBL4126094 0.81 NAMPT (0.35) NAMPTALDH1A1TBXAS1
SCHEMBL3650556 0.81 NAMPT (0.35) GPBAR1NAMPTCYP2C9PIK3CDPIK3CA
SCHEMBL4126083 0.80 GPBAR1 (0.36) GPBAR1NAMPTALDH1A1LMNAHTT
Fumaric Acid SCHEMBL3650347 0.79 TBXAS1 (0.36) NAMPTALDH1A1LMNAHTTNPSR1
Fumaric Acid SCHEMBL3650341 0.79 TBXAS1 (0.36) NAMPTALDH1A1LMNAHTTNPSR1
SCHEMBL3645990 0.79 PTGER2 (0.35) ABCC9ABCC8KCNJ11KCNJ8GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed