SCHEMBL3648437

SCHEMBL3648437

CC(C)(C)C(Cc1cc(-c2cccnc2Cl)c(S(=O)(=O)c2cccnc2)s1)NC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.36
MCL1 Q07820 1/20 0.35
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
KCNJ8 Q15842 1/20 0.35
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
AGTR2 P50052 3/20 0.33
ADAM17 P78536 1/20 0.33
SLC40A1 Q9NP59 1/20 0.32
HIF1A Q16665 1/20 0.32
ITGAV P06756 1/20 0.32
ALPL P05186 1/20 0.32
CKS1B P61024 1/20 0.32
SKP2 Q13309 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3650556 0.93 NAMPT (0.35) GPBAR1AGTR2SLC40A1EGFR
SCHEMBL3645989 0.88 ABCC9 (0.35) GPBAR1MCL1ABCC9ABCC8KCNJ11
SCHEMBL3799194 0.87 ABCC9 (0.35) MCL1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3803071 0.83 KDM4E (0.33) MCL1AGTR2
SCHEMBL3654308 0.81 SLC22A12 (0.33) GPBAR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3652836 0.81 AGTR2 (0.34) ABCC9ABCC8KCNJ11KCNJ8AGTR2
SCHEMBL3654949 0.81 AGTR2 (0.33) GPBAR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4130748 0.81 POLB (0.36) GPBAR1SLC40A1CKS1BSKP2ITGB3
SCHEMBL3806158 0.80 AGTR2 (0.32) MCL1AGTR2
SCHEMBL3653192 0.80 ABCC9 (0.36) GPBAR1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed