SCHEMBL3653192

SCHEMBL3653192

CC(C)(C)C(Cc1cc(S(=O)(=O)c2cccnc2)c(-c2cccnc2F)s1)NC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
FEN1 P39748 1/20 0.33
FPR1 P21462 1/20 0.33
NAMPT P43490 6/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
ITGAV P06756 1/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
PTGER2 P43116 2/20 0.32
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654495 0.91 ABCC9 (0.37) ABCC9ABCC8KCNJ11KCNJ8FPR1
SCHEMBL3645989 0.90 ABCC9 (0.35) ABCC9ABCC8KCNJ11KCNJ8NAMPT
SCHEMBL3649651 0.82 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8FPR1
SCHEMBL4126590 0.81 NAMPT (0.35) ABCC9ABCC8KCNJ11KCNJ8FEN1
SCHEMBL3648528 0.81 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8FEN1
SCHEMBL4126584 0.81 NAMPT (0.37) ABCC9ABCC8KCNJ11KCNJ8FEN1
SCHEMBL3652974 0.80 CYP2A6 (0.39) ABCC9ABCC8KCNJ11KCNJ8FEN1
SCHEMBL3648437 0.80 GPBAR1 (0.36) ABCC9ABCC8KCNJ11KCNJ8FPR1
Fumaric Acid SCHEMBL3651794 0.79 TBXAS1 (0.36) ABCC9ABCC8KCNJ11KCNJ8NAMPT
SCHEMBL3653193 0.79 PTGER2 (0.35) ABCC9ABCC8KCNJ11KCNJ8FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed