SCHEMBL3650244

SCHEMBL3650244

Cc1c(CC(NC(=O)O)C(C)(C)C)sc(S(=O)(=O)c2ccccc2)c1Br

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
ABCC9 O60706 2/20 0.33
ABCC8 Q09428 2/20 0.33
KCNJ11 Q14654 2/20 0.33
KCNJ8 Q15842 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
ATM Q13315 1/20 0.33
ANXA2 P07355 1/20 0.32
S100A10 P60903 1/20 0.32
THRB P10828 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL3648906 0.98 ANXA2 (0.33) MEN1KMT2AABCC9ABCC8KCNJ11
SCHEMBL3654646 0.80 ABCC9 (0.34) MEN1KMT2AABCC9ABCC8KCNJ11
Carbamic Acid SCHEMBL3651236 0.80 CA2 (0.35) MEN1KMT2AABCC9ABCC8KCNJ11
Hydrochloric Acid SCHEMBL3649320 0.76 CA12 (0.32) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4134961 0.75 GAA (0.38) ANXA2S100A10THRBALDH1A1GAA
SCHEMBL3650248 0.73 L3MBTL1 (0.34) MEN1KMT2AANXA2S100A10SMN1; SMN2
Hydrochloric Acid SCHEMBL3649181 0.73 LIPG (0.31) MEN1KMT2AMMP9MMP13CYP2C9
Carbamic Acid SCHEMBL3648907 0.72 HTT (0.34) MEN1KMT2AANXA2S100A10SMN1; SMN2
SCHEMBL3650241 0.72 HTR2C (0.38) MEN1KMT2ASMN1; SMN2GAAMAPT
SCHEMBL3653515 0.70 CA12 (0.35) KMT2AABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed