SCHEMBL3650696

SCHEMBL3650696

CC(C)(C)C(Cc1cc(Sc2cccnc2)c(Br)s1)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
PIK3CG P48736 1/20 0.35
PKM P14618 1/20 0.32
SLC8A1 P32418 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ITGB3 P05106 2/20 0.31
ITGAV P06756 2/20 0.31
ITGA2B P08514 2/20 0.31
CYP3A4 P08684 5/20 0.31
ECE1 P42892 1/20 0.31
TBXAS1 P24557 2/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649651 0.78 ABCC9 (0.39) ITGB3ITGAVITGA2B
SCHEMBL4132086 0.77 SMN1; SMN2 (0.37) PIK3CAPIK3CGNPC1RAB9AALDH1A1
SCHEMBL3650699 0.75 NR1D1 (0.32) PIK3CAPIK3CGNPC1RAB9ATBXAS1
SCHEMBL4132076 0.75 LMNA (0.37) PIK3CAPIK3CGPKMNPC1RAB9A
SCHEMBL3652851 0.74 POLB (0.34)
SCHEMBL3649825 0.72 DYRK1A (0.34)
SCHEMBL3650678 0.70 EDNRA (0.40) ALDH1A1
SCHEMBL3799194 0.70 ABCC9 (0.35) ITGB3ITGAVITGA2B
SCHEMBL3799450 0.69 CYP26A1 (0.34) ALDH1A1
SCHEMBL4023651 0.69 DYRK1A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed