SCHEMBL3652008

SCHEMBL3652008

Cc1ccc(S(=O)(=O)OC[C@H](C)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.51
LMNA P02545 1/20 0.49
ATM Q13315 1/20 0.49
CA2 P00918 5/20 0.48
CA5A P35218 2/20 0.48
GAA P10253 1/20 0.47
CA1 P00915 5/20 0.47
CTSK P43235 1/20 0.47
MAPT P10636 1/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3652010 1.00 P2RX7 (0.51) P2RX7LMNAATMCA2CA5A
SCHEMBL22552853 1.00 P2RX7 (0.51) P2RX7LMNAATMCA2CA5A
SCHEMBL3957822 0.87 P2RX7 (0.54) P2RX7LMNACTSK
SCHEMBL7100122 0.86 P2RX7 (0.49) P2RX7LMNAATMCA2CA1
SCHEMBL4972042 0.86 P2RX7 (0.54) P2RX7LMNACA5ACTSK
SCHEMBL6135399 0.86 P2RX7 (0.49) P2RX7LMNAATMCA2CA1
SCHEMBL9476901 0.86 CTRB1 (0.56) P2RX7LMNACA2GAACA1
SCHEMBL3948746 0.86 P2RX7 (0.54) P2RX7LMNACA5ACTSK
SCHEMBL7100119 0.86 P2RX7 (0.49) P2RX7LMNAATMCA2CA1
SCHEMBL7990303 0.85 P2RX7 (0.47) P2RX7LMNAATMCA2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2195288-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2010-06-16 EP disclosed
WO-2009036996-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2009-03-26 WO disclosed