SCHEMBL9476901

SCHEMBL9476901

Cc1ccc(S(=O)(=O)OC[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.56
P2RX7 Q99572 10/20 0.54
CTSL P07711 2/20 0.52
LMNA P02545 1/20 0.47
CTSK P43235 1/20 0.46
GAA P10253 1/20 0.46
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14370506 0.93 P2RX7 (0.55) CTRB1P2RX7CTSLCTSKCA1
SCHEMBL3070245 0.89 P2RX7 (0.48) CTRB1P2RX7CTSLLMNACA1
SCHEMBL7990303 0.87 P2RX7 (0.47) CTRB1P2RX7CTSLLMNACTSK
SCHEMBL7990292 0.86 LMNA (0.48) CTRB1P2RX7LMNACA1CA2
SCHEMBL3652008 0.86 P2RX7 (0.51) P2RX7LMNACTSKGAACA1
SCHEMBL22552853 0.86 P2RX7 (0.51) P2RX7LMNACTSKGAACA1
SCHEMBL3652010 0.86 P2RX7 (0.51) P2RX7LMNACTSKGAACA1
SCHEMBL27447522 0.86 CTRB1 (0.55) CTRB1P2RX7CTSLCTSKGAA
SCHEMBL1258429 0.86 ATM (0.56) P2RX7CTSLLMNACTSKGAA
SCHEMBL1258432 0.86 ATM (0.56) P2RX7CTSLLMNACTSKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5244905-A Gastric antisecretory, antipsychotic, appetite suppressants WARNER-LAMBERT COMPANY (US) 1993-09-14 US disclosed
WO-1992004348-A1 N-SUBSTITUTED CYCLOALKYL AND POLYCYCLOAKYL POLYHYDRO-Β-CARBOLINE-PHENYLALANINE-AND PHENETHYLAMINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1992-03-19 WO disclosed