SCHEMBL3653449

SCHEMBL3653449

COCCn1ccc2cc(N)ccc21

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.54
GLO1 Q04760 2/20 0.47
HTR2C P28335 6/20 0.43
EGFR P00533 1/20 0.43
BRPF1 P55201 1/20 0.42
NTSR1 P30989 1/20 0.42
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
HTR2A P28223 5/20 0.39
HTR6 P50406 1/20 0.39
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4277776 0.86 PRKCI (0.46) PRKCIGLO1HTR2CEGFRBRPF1
SCHEMBL3650822 0.81 PRKCI (0.59) PRKCIHTR2CEGFRBRPF1NTSR1
SCHEMBL31735936 0.81 GLO1 (0.46) GLO1HTR2CPLGPLAUMTNR1A
SCHEMBL27593312 0.81 PRKCI (0.47) PRKCIGLO1EGFRBRPF1NTSR1
SCHEMBL1612942 0.81 HTR2C (0.55) GLO1HTR2CNTSR1MTNR1AMTNR1B
SCHEMBL5333977 0.81 HTR2C (0.55) GLO1HTR2CMTNR1AMTNR1BHTR2A
SCHEMBL21051475 0.81 GLO1 (0.50) GLO1HTR2CPLGPLAUMTNR1A
SCHEMBL6789563 0.80 PRKCI (0.56) PRKCIHTR2CEGFRBRPF1NTSR1
SCHEMBL14117445 0.79 GLO1 (0.46) GLO1HTR2CPLGPLAUMTNR1A
SCHEMBL5089820 0.79 PRKCI (0.56) PRKCIHTR2CEGFRBRPF1NTSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115768771-A Arylsulfonyl derivatives and their use as muscarinic acetylcholine receptor M5 inhibitors 范德堡大学 2023-03-07 CN claimed
EP-2197875-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2010-06-23 EP claimed
WO-2009037222-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS VIA PHARMACEUTICALS, INC. (US) 2009-03-26 WO claimed
WO-2025245461-A1 METHODS OF ACTIVATING FOXN1 THYMOFOX INC. (US) 2025-11-27 WO disclosed
WO-2025245484-A1 FOXN1 ACTIVATORS THYMOFOX INC. (US) 2025-11-27 WO disclosed
CN-117486865-A Pyrimidine derivatives as kinase inhibitors 艾森医药公司 2024-02-02 CN disclosed
CN-112592334-B Pyrimidine derivatives as kinase inhibitors 艾森医药公司 2023-10-27 CN disclosed
CN-115768771-A Arylsulfonyl derivatives and their use as muscarinic acetylcholine receptor M5 inhibitors 范德堡大学 2023-03-07 CN disclosed
CN-112592334-A Pyrimidine derivatives as kinase inhibitors 艾森生物科学公司 2021-04-02 CN disclosed
US-10562918-B2 Heterocyclic compounds and uses thereof ACEA Therapeutics, Inc. (US) 2020-02-18 US disclosed
US-10562918-B2 Heterocyclic compounds and uses thereof ACEA Therapeutics, Inc. (US) 2020-02-18 US disclosed
US-9464089-B2 Heterocyclic compounds and uses thereof ACEA BIOSCIENCES INC. (US) 2016-10-11 US disclosed
US-9464089-B2 Heterocyclic compounds and uses thereof ACEA BIOSCIENCES INC. (US) 2016-10-11 US disclosed
CN-105916851-A Pyrimidine derivatives as kinase inhibitors 艾森生物科学公司 2016-08-31 CN disclosed
US-20150133457-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA BIOSCIENCES INC. 2015-05-14 US disclosed
US-20150133457-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA BIOSCIENCES INC. 2015-05-14 US disclosed
US-20150133457-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA BIOSCIENCES INC. 2015-05-14 US disclosed
WO-2015006754-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF ACEA BIOSCIENCES INC. (US) 2015-01-15 WO disclosed
EP-2197875-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2010-06-23 EP disclosed
WO-2009037222-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS VIA PHARMACEUTICALS, INC. (US) 2009-03-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150133457-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF BMX, BLK, BTK PRKCI 1307/4885GLO1 3350/4885HTR2C 1627/4885
US-10562918-B2 Heterocyclic compounds and uses thereof BMX, BLK, BTK PRKCI 1307/4885GLO1 3350/4885HTR2C 1627/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.