SCHEMBL365476

SCHEMBL365476

CS(=O)(=O)NC(=O)c1ccc2cc3ccccc3n2c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.46
SCN2B O60939 8/20 0.46
SCN1B Q07699 8/20 0.46
SCN5A Q14524 7/20 0.46
SCN1A P35498 6/20 0.46
CCR2 P41597 1/20 0.43
MYC P01106 2/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
HTR3A P46098 1/20 0.42
PPARG P37231 1/20 0.41
PTPN1 P18031 1/20 0.41
MCL1 Q07820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366724 0.79 CHRNA7 (0.43) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL365475 0.78 SCN9A (0.48) SCN9ASCN2BSCN1BSCN5ASCN1A
SCHEMBL6851185 0.76 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL366784 0.72 SCN9A (0.50) SCN9ASCN2BSCN1BSCN5ASCN1A
SCHEMBL366354 0.70 SCN9A (0.46) SCN9ASCN2BSCN1BSCN5ASCN1A
SCHEMBL6412569 0.69 CHRNA7 (0.84) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL6417457 0.68 CHRNA7 (0.49) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL364110 0.68 HDAC3 (0.58) SCN9ASCN2BSCN1BSCN5ASCN1A
SCHEMBL28531553 0.67 CHRNA7 (0.51) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL366978 0.67 SCN9A (0.45) SCN9ASCN2BSCN1BSCN5ASCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed