SCHEMBL3655686

SCHEMBL3655686

C=Cc1ncc(C(=O)O)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.43
NAPRT Q6XQN6 1/20 0.43
TTR P02766 1/20 0.42
TSHR P16473 1/20 0.41
MGAM O43451 1/20 0.39
HCAR3 P49019 1/20 0.37
P4HA1 P13674 2/20 0.37
P4HTM Q9NXG6 2/20 0.37
SRD5A2 P31213 1/20 0.37
PLAU P00749 1/20 0.37
TPMT P51580 2/20 0.36
MIF P14174 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649983 0.80 MGAM (0.40) HCAR2NAPRTMGAMHCAR3P4HA1
SCHEMBL16616328 0.80 MGAM (0.40) HCAR2NAPRTMGAMHCAR3P4HA1
SCHEMBL1424865 0.77 STAT3 (0.35) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL29365646 0.75 HCAR2 (0.50) HCAR2NAPRTTTRTSHRMGAM
SCHEMBL232290 0.75 HCAR2 (0.50) HCAR2NAPRTTTRTSHRMGAM
SCHEMBL25396560 0.75 RORC (0.36) ALDH1A1KDM4EPOLBMEN1LMNA
SCHEMBL199221 0.73 TTR (0.54) HCAR2NAPRTTTRTSHRMGAM
Hydrochloric Acid SCHEMBL7476482 0.73 HCAR2 (0.48) HCAR2NAPRTTTRTSHRMGAM
SCHEMBL3650453 0.73 HCAR2 (0.48) HCAR2NAPRTTTRTSHRMGAM
SCHEMBL30821436 0.73 PDXK (0.36) TTRHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101522670-B Pyridin-3-yl derivatives as immunomodulators ACTELION PHARMACEUTICALS LTD 2012-05-23 CN disclosed
EP-2195311-A1 PYRIDINE DERIVATIVES AS S1P1/EDG1 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd. (CH) 2010-06-16 EP disclosed
CN-101522670-A Pyridin-3-yl derivatives as immunomodulators ACTELION PHARMACEUTICALS LTD (CH) 2009-09-02 CN disclosed
WO-2009024905-A1 PYRIDINE DERIVATIVES AS S1P1/EDG1 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2009-02-26 WO disclosed