SCHEMBL3656136

SCHEMBL3656136

Oc1ccccc1-n1ncc2cc(CC(c3ccc(Cl)cc3Cl)C(O)C(F)(F)F)ccc21

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMO Q99835 9/20 0.35
PDE9A O76083 1/20 0.35
HDAC8 Q9BY41 1/20 0.33
KCNH2 Q12809 1/20 0.33
NR3C1 P04150 3/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
TP53 P04637 1/20 0.32
SCN9A Q15858 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658449 0.85 NR3C1 (0.41) SMONR3C1CYP11B1CYP11B2
SCHEMBL3659346 0.85 NR3C1 (0.38) SMONR3C1CYP11B1CYP11B2
SCHEMBL837360 0.75 NR3C1 (0.43) NR3C1CYP11B1CYP11B2SCN9A
SCHEMBL1414860 0.69 NR3C1 (0.42) NR3C1CYP11B1CYP11B2TP53SCN9A
SCHEMBL1414583 0.67 ADRA2C (0.31)
SCHEMBL3658681 0.67 MAPT (0.32) KCNH2
SCHEMBL3660501 0.64 MAPT (0.32)
SCHEMBL838615 0.64 NR3C1 (0.43) SMONR3C1CYP11B1CYP11B2SCN9A
SCHEMBL837940 0.63 NR3C1 (0.51) NR3C1CYP11B1CYP11B2
SCHEMBL838977 0.62 SMO (0.43) SMONR3C1CYP11B1CYP11B2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP claimed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO claimed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed