SCHEMBL3658449

SCHEMBL3658449

Oc1ccc(-n2ncc3cc(CC(c4ccc(Cl)cc4Cl)C(O)C(F)(F)F)ccc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 10/20 0.41
SMO Q99835 9/20 0.41
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3659346 0.90 NR3C1 (0.38) NR3C1SMOCYP11B1CYP11B2PGR
SCHEMBL3656136 0.85 SMO (0.35) NR3C1SMOCYP11B1CYP11B2
SCHEMBL837594 0.73 NR3C1 (0.51) NR3C1CYP11B1CYP11B2
SCHEMBL1414583 0.68 ADRA2C (0.31)
SCHEMBL3658681 0.68 MAPT (0.32)
SCHEMBL1415502 0.67 NR3C1 (0.48) NR3C1CYP11B1CYP11B2
SCHEMBL3659001 0.65 TDP1 (0.40)
SCHEMBL3660501 0.65 MAPT (0.32)
SCHEMBL4282965 0.64 NR3C1 (0.86) NR3C1CYP11B1CYP11B2PGR
SCHEMBL837940 0.64 NR3C1 (0.51) NR3C1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP claimed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO claimed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed