SCHEMBL3659346

SCHEMBL3659346

Oc1cccc(-n2ncc3cc(CC(c4ccc(Cl)cc4Cl)C(O)C(F)(F)F)ccc32)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 7/20 0.38
PGR P06401 1/20 0.38
HPGD P15428 1/20 0.36
SMO Q99835 9/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
TRPV1 Q8NER1 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658449 0.90 NR3C1 (0.41) NR3C1PGRSMOCYP11B1CYP11B2
SCHEMBL3656136 0.85 SMO (0.35) NR3C1SMOCYP11B1CYP11B2
SCHEMBL838520 0.74 NR3C1 (0.48) NR3C1PGRHPGDCYP11B1CYP11B2
SCHEMBL1415940 0.69 NR3C1 (0.46) NR3C1PGRHPGDCYP11B1CYP11B2
SCHEMBL3658681 0.66 MAPT (0.32)
SCHEMBL1414583 0.66 ADRA2C (0.31)
SCHEMBL27074837 0.65 NR3C1 (0.59) NR3C1PGRHPGDCYP11B2MAPK8
SCHEMBL838181 0.64 NR3C1 (0.47) NR3C1PGRSMOCYP11B1CYP11B2
SCHEMBL837940 0.64 NR3C1 (0.51) NR3C1CYP11B1CYP11B2
SCHEMBL838199 0.64 NR3C1 (0.44) NR3C1PGRHPGDSMOCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP claimed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO claimed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed